Nonpeptidic HIV protease inhibitors: 6-alkyl-5, 6-dihydropyran-2-ones possessing achiral 3-(4-amino/carboxamide-2-t-butyl, 5-methylphenyl thio) moiety: Antiviral activities and pharmacokinetic properties

J. V. N. Vara Prasad(Pfizer (United States)), Joanne Brodfuehrer(Pfizer (United States)), Fred E. Boyer(Warde Medical Laboratory), Larry J. Markoski(Pfizer (United States)), Christopher Gajda(Pfizer (United States)), K. R. Krishna Iyer(University of Michigan), Susan E. Hagen(Pfizer (United States)), Elizabeth A. Lunney(Pfizer (United States)), Edmund L. Ellsworth(Pfizer (United States)), Peter J. Tummino(Ensemble Therapeutics (United States)), James M. Saunders(Pfizer (United States)), Carolyn Nouhan(Pfizer (United States)), Michael Sinz(Rutgers, The State University of New Jersey), Donna Ferguson(Pfizer (United States)), Donald Hupe(Pfizer (United States)), Steven VanderRoest(Pfizer (United States)), Bradley D. Tait(Pfizer (United States)), Stephen J. Gracheck(Pfizer (United States)), John M. Domagala(Pfizer (United States)), Tod P. Holler(Pfizer (United States))
Bioorganic & Medicinal Chemistry Letters
June 1, 1999
Cited by 8


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