Bioactivation of a Novel 2-Methylindole-Containing Dual Chemoattractant Receptor-Homologous Molecule Expressed on T-Helper Type-2 Cells/d-Prostanoid Receptor Antagonist Leads to Mechanism-Based CYP3A Inactivation: Glutathione Adduct Characterization and Prediction of In Vivo Drug-Drug Interaction
Simon Wong, Bradley K. Wong(United States Military Academy), Michelle Tadano Lohr, Kirk R. Henne(Denali Therapeutics (United States)), Michael G. Johnson(University of California, Berkeley), Peter W. Fan, George Tonn, Raju Subramanian(Gilead Sciences (United States))
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