Substrate-Assisted Inhibition of Ubiquitin-like Protein-Activating Enzymes: The NEDD8 E1 Inhibitor MLN4924 Forms a NEDD8-AMP Mimetic In Situ

James E. Brownell(Millennium Engineering and Integration (United States)), Michael D. Sintchak(Millennium Engineering and Integration (United States)), James M. Gavin(Millennium Engineering and Integration (United States)), Hua Liao(Millennium Engineering and Integration (United States)), Frank J. Bruzzese(Millennium Engineering and Integration (United States)), Nancy J. Bump(Millennium Engineering and Integration (United States)), Teresa A. Soucy(Millennium Engineering and Integration (United States)), Michael A. Milhollen(Millennium Engineering and Integration (United States)), Xiaofeng Yang(Millennium Engineering and Integration (United States)), Anne L. Burkhardt(Millennium Engineering and Integration (United States)), Jingya Ma(Millennium Engineering and Integration (United States)), Huay-Keng Loke(Millennium Engineering and Integration (United States)), Trupti Lingaraj(Millennium Engineering and Integration (United States)), Dongyun Wu(Millennium Engineering and Integration (United States)), Kristin B. Hamman(Millennium Engineering and Integration (United States)), James J. Spelman(Millennium Engineering and Integration (United States)), Courtney Cullis(Millennium Engineering and Integration (United States)), Steven Langston(Millennium Engineering and Integration (United States)), Štěpán Vyskočil(Millennium Engineering and Integration (United States)), Todd B. Sells(Millennium Engineering and Integration (United States)), William D. Mallender(Millennium Engineering and Integration (United States)), Irache Visiers(Millennium Engineering and Integration (United States)), Ping Li(Millennium Engineering and Integration (United States)), Christopher F. Claiborne(Millennium Engineering and Integration (United States)), Mark Rolfe(Millennium Engineering and Integration (United States)), Joseph B. Bolen(Millennium Engineering and Integration (United States)), Lawrence R. Dick(Millennium Engineering and Integration (United States))
Molecular Cell
January 1, 2010
Cited by 461Open Access
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