Discovery of Pyrophosphate Diesters as Tunable, Soluble, and Bioorthogonal Linkers for Site-Specific Antibody–Drug ConjugatesJeffrey C. Kern, R. M. Garbaccio, Anthony Palmieri et al.|Journal of the American Chemical Society|2016Cited by 141
Novel Phosphate Modified Cathepsin B Linkers: Improving Aqueous Solubility and Enhancing Payload Scope of ADCsJeffrey C. Kern, R. M. Garbaccio, Philip E. Brandish et al.|Bioconjugate Chemistry|2016Cited by 94