Novel Phosphate Modified Cathepsin B Linkers: Improving Aqueous Solubility and Enhancing Payload Scope of ADCs

Jeffrey C. Kern, R. M. Garbaccio(United States Military Academy), Rena Zhang, Nick Knudsen(Ambrx (United States)), Mangeng Cheng, Anthony Manibusan(Ambrx (United States)), Juhi Firdos(Ambrx (United States)), Damien Bresson(Ambrx (United States)), Guo Feng, Linda Liang(Merck & Co., Inc., Rahway, NJ, USA (United States)), Andrew H. Beck(Brown University), Ying Sun(Torrey Pines Institute For Molecular Studies), Philip E. Brandish(Merck & Co., Inc., Rahway, NJ, USA (United States)), Dennis Gately(Ambrx (United States)), Deborah Dooney
Bioconjugate Chemistry
July 29, 2016
Cited by 94


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