Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer
Steven Langston(Takeda (United States)), Xiaofeng Yang(Millennium Engineering and Integration (United States)), Neil Bence(Nurix (United States)), Christopher F. Claiborne(Millennium Engineering and Integration (United States)), Anya Lublinsky(Takeda (United States)), Ryan Chau(Takeda (United States)), William D. Mallender(Millennium Engineering and Integration (United States)), Nitya Durvasula(Takeda (United States)), Bei-Ching Chuang(Takeda (United States)), James Minissale(Takeda (United States)), Katherine Galvin(Takeda (United States)), Scott Weston Lane(Takeda (United States)), Larry S. Cohen(Takeda (United States)), Vaishali Shindi(Takeda (United States)), Koji Ono(Takeda (Japan)), Yana Wang(Takeda (United States)), Shumet Hailu(Takeda (United States)), Paul D. Greenspan(Takeda (United States)), Misook Kim(Takeda (United States)), Nanda K. Gulavita(Takeda (United States)), Michael D. Sintchak(Millennium Engineering and Integration (United States)), David Lok(Takeda (United States)), Stephen Grossman(Takeda (United States)), He N. Xu(Takeda (United States)), Charles McIntyre(Takeda (United States)), Ashok D. Patil(Takeda (United States)), Nina Molchinova(Takeda (United States)), Jianping Guo(Sun Yat-sen University), Teresa A. Soucy(Millennium Engineering and Integration (United States)), Melissa Gallery(Takeda (United States)), Zhigen Hu(Takeda (United States)), Matthew O. Duffey(Takeda (United States)), Kelly Connolly(Takeda (United States)), Kara M. Hoar(Takeda (United States)), Jessica Grieves(Takeda (United States)), Roushan Afroze(Takeda (United States)), Xingyue He(Takeda (United States)), Mitsuhiro Ito(Takeda (Japan)), Hirotake Mizutani(Millennium Engineering and Integration (United States)), Jeffrey Gaulin(Millennium Engineering and Integration (United States)), Jessica Riceberg(Takeda (United States)), Dylan B. England(Takeda (United States)), Douglas Bowman(Takeda (United States)), Rachel E. Gershman(Millennium Engineering and Integration (United States)), Miho Mizutani(Takeda (United States)), Keli Song(Takeda (United States)), Yongbo Hu(Takeda (United States)), Scott Freeze(Takeda (United States)), Nancy J. Bump(Millennium Engineering and Integration (United States)), Mark G. Qian(Takeda (United States))
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