Synthesis of 5,6-Dihydro-4-hydroxy-2- pyrones as HIV-1 Protease Inhibitors:  The Profound Effect of Polarity on Antiviral Activity

Susan E. Hagen(Pfizer (United States)), Steven VanderRoest(Pfizer (United States)), Harriet W. Hamilton(Pfizer (United States)), Larry J. Markoski(Pfizer (United States)), Christopher Gajda(Pfizer (United States)), Elizabeth A. Lunney(Pfizer (United States)), Edmund L. Ellsworth(Pfizer (United States)), Peter J. Tummino(Intarcia Therapeutics (United States)), James M. Saunders(Pfizer (United States)), Carolyn Nouhan(Pfizer (United States)), Donna Ferguson(Pfizer (United States)), Donald Hupe(Pfizer (United States)), J. V. N. Vara Prasad(Pfizer (United States)), F Boyer(Pfizer (United States)), Bradley D. Tait(Pfizer (United States)), Stephen J. Gracheck(Pfizer (United States)), John M. Domagala(Pfizer (United States)), Bruce A. Steinbaugh(Pfizer (United States))
Journal of Medicinal Chemistry
November 1, 1997
Cited by 62


Related Papers