Identification and Characterization of 4-Methylbenzyl 4-[(Pyrimidin-2-ylamino)methyl]piperidine-1-carboxylate, an Orally Bioavailable, Brain Penetrant NR2B Selective<i>N</i>-Methyl-<scp>d</scp>-Aspartate Receptor Antagonist

Nigel J. Liverton(United States Military Academy), Kenneth S. Koblan(Sumitomo Dainippon Pharma (United States)), Stanley L. Gaul(United States Military Academy), John A. McCauley(Fox Chase Cancer Center), Christopher F. Claiborne(Roche (Switzerland)), David A. Claremon, Anthony G. DiLella(United States Military Academy), Bohumil Bednár̂(Institute of Chemical Technology), John W. Butcher(United States Military Academy), Rodney A. Bednar(United States Military Academy), Joseph J. Lynch(United States Military Academy), Brian E. Libby(United States Military Academy), Gary L. Stump(United States Military Academy), Hao Wang(Tongji University), Kevin T. Nguyen(Navidea Biopharmaceuticals (United States)), Scott D. Mosser(United States Military Academy), Elizabeth A. Lyle, Michael E. Cunningham(Children's National), James A. Yergey, Hong Sun(United States Military Academy)
Journal of Medicinal Chemistry
January 24, 2007
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