Using the Golden Triangle to optimize clearance and oral absorptionTed W. Johnson, Martin P. Edwards, Klaus Dress|Bioorganic & Medicinal Chemistry Letters|2009Cited by 382
The development and SAR of pyrrolidine carboxamide 11β-HSD1 inhibitorsHengmiao Cheng, Paul A. Rejto, Bridget Cole et al.|Bioorganic & Medicinal Chemistry Letters|2010Cited by 44
Discovery of PF-07265028, A Selective Small Molecule Inhibitor of Hematopoietic Progenitor Kinase 1 (HPK1) for the Treatment of CancerRebecca A. Gallego, Sajiv K. Nair, Sujin Cho-Schultz et al.|Journal of Medicinal Chemistry|2024Cited by 19
N-(Pyridin-2-yl) arylsulfonamide inhibitors of 11β-hydroxysteroid dehydrogenase type 1: Strategies to eliminate reactive metabolitesSajiv K. Nair, Deepak Dalvie, Jean Matthews et al.|Bioorganic & Medicinal Chemistry Letters|2013Cited by 11
Discovery of Atirmociclib (PF-07220060): A Potent and Selective CDK4 InhibitorGary M. Gallego, Sajiv K. Nair, Cynthia L. Palmer et al.|Journal of Medicinal Chemistry|2025Cited by 4