Discovery of Atirmociclib (PF-07220060): A Potent and Selective CDK4 Inhibitor

Gary M. Gallego(Theravance Biopharma (United States)), Sajiv K. Nair(Pfizer (United States)), Sacha Ninkovic(Pfizer (United States)), Louise Bernier(Pfizer (United States)), Julie Cianfrogna(Pfizer (United States)), John C. Kath(Pfizer (United States)), Lars Anders(Pfizer (United States)), Robert S. Kania(RG Biopharma (United States)), Aida Sacaan(Pfizer (United States)), Loretta M. Cox(Pfizer (United States)), Bernadette Pascual(Pfizer (United States)), Na Wei(Pfizer (United States)), Lisa D. Marroquin(Pfizer (United States)), Judith G. Deal(Pfizer (United States)), Britton Boras(Pfizer (United States)), Martin P. Edwards(Pfizer (United States)), Mehran Jalaie(Pfizer (United States)), Neal W. Sach(Pfizer (United States)), Sujin Cho-Schultz(Pfizer (United States)), Casey L. Quinlan(Pfizer (United States)), Suvi T. M. Orr(Tracon Pharmaceuticals (United States)), Fengjuan Cao(Pfizer (United States)), Klaus Dress(Pfizer (United States)), Eric F. Johnson(Pfizer (United States)), Hong Shen(Pfizer (United States)), Cynthia L. Palmer(Pfizer (United States)), Ping Chen(Shandong Jiaotong University), Jennifer Lafontaine(Pfizer (United States)), Matthew D. Petroski(Pfizer (United States))
Journal of Medicinal Chemistry
December 5, 2025
Cited by 4


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