Discovery of a Selective Series of Inhibitors of <i>Plasmodium falciparum</i> HDACsJesus M. Ontoria, Steven J. Harper, Ottavia Cecchetti et al.|ACS Medicinal Chemistry Letters|2016Cited by 42
Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and BenzamidesAlberto Bresciani, Steven J. Harper, Jesus M. Ontoria et al.|ACS Medicinal Chemistry Letters|2018Cited by 32
Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 InteractionJesus M. Ontoria, Steven J. Harper, Ilaria Biancofiore et al.|ACS Medicinal Chemistry Letters|2020Cited by 29
SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 proteaseStefania Colarusso, Jesus M. Ontoria, Federica Ferrigno et al.|Bioorganic & Medicinal Chemistry|2022Cited by 11
Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitroFederica Ferrigno, Jesus M. Ontoria, Ilaria Biancofiore et al.|Bioorganic & Medicinal Chemistry Letters|2018Cited by 5