Discovery of a Selective Series of Inhibitors of <i>Plasmodium falciparum</i> HDACsJesus M. Ontoria, Steven J. Harper, Ralph Laufer et al.|ACS Medicinal Chemistry Letters|2016Cited by 42
Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and BenzamidesAlberto Bresciani, Steven J. Harper, Jesus M. Ontoria et al.|ACS Medicinal Chemistry Letters|2018Cited by 32
Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 InteractionJesus M. Ontoria, Steven J. Harper, Ilaria Biancofiore et al.|ACS Medicinal Chemistry Letters|2020Cited by 29
Identification of a series of 4-[3-(quinolin-2-yl)-1,2,4-oxadiazol-5-yl]piperazinyl ureas as potent smoothened antagonist hedgehog pathway inhibitorsJesus M. Ontoria, Philip Jones, Laura Llauger Bufi et al.|Bioorganic & Medicinal Chemistry Letters|2011Cited by 28
N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxamides as highly potent smoothened antagonistsEster Muraglia, Philip Jones, Jesus M. Ontoria et al.|Bioorganic & Medicinal Chemistry Letters|2011Cited by 25