Site-Directed Mutagenesis and Time-Resolved Fluorescence Spectroscopy Reveal That Two Hydrogen-Bonded Carboxylic Side Chains Are Essential for GPR68 Proton Sensing and G Protein Binding

B.M. Kapur(Boehringer Ingelheim (Germany)), Gisela Schnapp(Boehringer Ingelheim (Germany)), Ana‐Nicoleta Bondar(Forschungszentrum Jülich), Eva M. Garrido‐Martín(Boehringer Ingelheim (Germany)), Herbert Nar(Boehringer Ingelheim (Germany)), Esther Schmidt(European Bioinformatics Institute), Michael Schuler(Boehringer Ingelheim (Germany))
ACS Pharmacology & Translational Science
October 17, 2025
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