Accelerating Medicinal Chemistry: A C(sp3)-rich Fragment Toolbox for Redox-Neutral Cross-Coupling

Jet Tsien(Scripps Research Institute), Phil S. Baran(Scripps Research Institute), Áron Péter(University of Manchester), Johnny W. Lee(Pfizer (United States)), Michael R. Collins(Pfizer (United States)), Baiyang Jiang(Scripps Research Institute), Shuanghu Wang, Philippe N. Bolduc(Biogen (United States)), Megan A. Emmanuel(Siemens (Hungary)), Yu Kawamata(Scripps Research Institute), Xin Zheng(Union Hospital), Jennifer X. Qiao(Princeton University), Martins S. Oderinde(Bristol-Myers Squibb (United States)), Martin Bravo(Pfizer (United States)), Michael C. Nicastri(Biogen (United States)), Shalini Dey(Biogen (United States)), Maximilian D. Palkowitz(Bristol-Myers Squibb (Germany))
ChemRxiv
May 12, 2025
Cited by 1


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