Discovery and Synthesis of GS-7682, a Novel Prodrug of a 4′-CN-4-Aza-7,9-Dideazaadenosine <i>C</i> -Nucleoside with Broad-Spectrum Potency Against Pneumo- and Picornaviruses and Efficacy in RSV-Infected African Green Monkeys

Dustin S. Siegel(Gilead Sciences (United States)), Richard L. Mackman(Gilead Sciences (United States)), Philip J. Kuehl, Bindu Goyal(Gilead Sciences (United States)), Ona Barauskas(Gilead Sciences (United States)), Hammad Irshad(Lovelace Medical Center), Hon C. Hui(Gilead Sciences (United States)), Edward Doerffler(Gilead Sciences (United States)), Davin Rautiola(Université Bourgogne Franche-Comté), Raju Subramanian(Gilead Sciences (United States)), Joy Y. Feng(Gilead Sciences (United States)), Hai Yang(Natural Resources Conservation Service), Kirsten M. Stray(Gilead Sciences (United States)), Gregory Chin, Bin Ma(Tongji University), Tomáš Cihlář(Gilead Sciences (United States)), Chris Palmiotti(Gilead Sciences (United States)), Adrian Tomkinson(Gilead Sciences (United States)), Minji Seung(Gilead Sciences (United States)), Michael O. Clarke(Gilead Sciences (United States)), Nicholas C. Riola(Gilead Sciences (United States)), Nani Kadrichu(Inspire), Michel Perron(Gilead Sciences (United States)), Arya Vijjapurapu(Gilead Sciences (United States)), Meghan S. Vermillion(Lovelace Respiratory Research Institute), A. Nayak(Gilead Sciences (United States)), Yili Xu(Yanshan University), John P. Bilello(Global Vaccines (United States)), Gary Lee(Sir Charles Gairdner Hospital), Jared Pitts(Gilead Sciences (United States)), Ting Wang(San Francisco Art Institute), Eisuke Murakami(Gilead Sciences (United States)), Kazuya Ishida(Gilead Sciences (United States)), Xiaofeng Zhao(Gilead Sciences (United States)), Bruno Marchand(Gilead Sciences (United States)), Michael Keeney(Mayo Clinic in Arizona), Scott Ellis(Gilead Sciences (United States)), Kwon Soo Chun(Gilead Sciences (United States)), Lijun Zhang(Dalian Medical University), Jason K. Perry(Pulmatrix (United States))
bioRxiv (Cold Spring Harbor Laboratory)
April 19, 2024
Cited by 0


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