Discovery of Thieno[2,3-d]pyrimidine-based KRAS G12D inhibitors as potential anticancer agents via combinatorial virtual screening

Ling Li(Tumor Hospital of Guangxi Medical University), Jianjun Chen(Southern Medical University), Bulian Deng(Southern Medical University), Ruiyao Mai(Southern Medical University), Jin Liu(Southern Medical University), Zichao Yang(Southern Medical University), Junli Huang(Academy of Medical Sciences), Huiting Zhao(Jiangsu University), Yichang Ren(Southern Medical University)
European Journal of Medicinal Chemistry
March 3, 2022
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