Trivalent PROTACs enhance protein degradation via combined avidity and cooperativity

Satomi Imaide(University of Dundee), Kristin M. Riching(Promega (United States)), Nikolai Makukhin(University of Dundee), Vesna Vetma(University of Dundee), Claire Whitworth(University of Dundee), Scott J. Hughes(University of Dundee), Nicole Trainor(University of Dundee), Sarah D. Mahan(Promega (United States)), Nancy E. Murphy(Promega (United States)), Angus D. Cowan(University of Dundee), Kwok-Ho Chan(University of Dundee), Conner Craigon(University of Dundee), Andrea Testa(University of Dundee), Chiara Maniaci(University of Dundee), Marjeta Urh(Promega (United States)), Danette L. Daniels(Promega (United States)), Alessio Ciulli(University of Dundee)
Nature Chemical Biology
October 21, 2021
Cited by 234Open Access
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