Discovery of novel 9-heterocyclyl substituted 9H-purines as L858R/T790M/C797S mutant EGFR tyrosine kinase inhibitors

Hao Lei(Xi'an Jiaotong University), San‐Qi Zhang(Xi'an Jiaotong University), Junjie Zhang(Chemical Synthesis Lab), Hao Zhang(Qingdao University), Yanjie Liu(Tongji University), Shu Fan(Xi'an Jiaotong University), Minhang Xin(Zhejiang University), Aqun Zheng(Xi'an Jiaotong University), Yuan‐Yuan Hei(Xi'an Jiaotong University)
European Journal of Medicinal Chemistry
November 16, 2019
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