Discovery of potent epidermal growth factor receptor (EGFR) degraders by proteolysis targeting chimera (PROTAC)

Hao Zhang(Affiliated Hospital of Jining Medical University), San‐Qi Zhang(Xi'an Jiaotong University), Minhang Xin(Xi'an Jiaotong University), Xiao-Xiao Xi(Xi'an Jiaotong University), Junjie Zhang(Chemical Synthesis Lab), Yanjie Liu(Harbin Medical University), Shuai Mao(Xi'an Jiaotong University), Axin Lu(Xi'an Jiaotong University), Hongyi Zhao(Xi'an Jiaotong University)
European Journal of Medicinal Chemistry
January 13, 2020
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