Functional TRIM24 degrader via conjugation of ineffectual bromodomain and VHL ligands

Lara Gechijian(Jnana Therapeutics (United States)), James E. Bradner(Novartis (China)), Jennifer A. Perry(Dana-Farber Cancer Institute), Joshiawa Paulk(Novartis (United States)), Nathanael S. Gray(Stanford University), Matthew A. Lawlor(Dana-Farber Cancer Institute), Jaime M. Reyes(Dana-Farber Cancer Institute), Georg E. Winter(CeMM Research Center for Molecular Medicine), Michael A. Erb(Scripps Research Institute), Hyuk‐Soo Seo(Dana-Farber Cancer Institute), Jun Qi(Georgia Institute of Technology), Mousheng Xu(Dana-Farber Cancer Institute), Dennis L. Buckley(Novartis (United States)), Nicholas Kwiatkowski(Woomera Therapeutics), Christopher J. Ott(Broad Institute), Sirano Dhe‐Paganon(University of Toronto), Thomas G. Scott(Dana-Farber Cancer Institute)
Nature Chemical Biology
March 5, 2018
Cited by 229


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