Diversity-oriented synthesis yields novel multistage antimalarial inhibitors

Nobutaka Kato(Broad Institute), Dyann F. Wirth(Harvard University), Matthias Marti(University of Zurich), Clemens H. M. Kocken(Biomedical Primate Research Centre), Jon Clardy(Harvard University), Jacob A. McPhail(University of Victoria), Manmohan Sharma(International Centre for Genetic Engineering and Biotechnology), Maurice A. Itoe(Harvard University), Gillian L. Dornan(University of Victoria), Sandra March(Broad Institute), Micah Maetani(Broad Institute), Morgane Sayes(Broad Institute), Paul A. Clemons(Broad Institute), Eamon Comer(Broad Institute), Timothy A. Lewis(Broad Institute), Jessica Bastien(Broad Institute), Sangeeta N. Bhatia(Broad Institute), Victoria Corey(University of California San Diego), Mathias J. Wawer(Broad Institute), Ping S. Lui(Harvard University), Arvind Sharma(International Centre for Genetic Engineering and Biotechnology), Flaminia Catteruccia(Howard Hughes Medical Institute), Michael A. Foley(Harvard University), Eli L. Moss(Broad Institute), Tomoyo Sakata‐Kato(Drug Discovery Laboratory (Norway)), Karin M. J. Koolen(TropIQ Health Sciences), Amit Sharma(International Centre for Genetic Engineering and Biotechnology), Vicky M. Avery(Griffith University), Joshua A. Bittker, David C. Clarke(Harvard University), Bennett C. Meier(Broad Institute), Daniel E. Neafsey(Broad Institute), Emily Lund(Harvard University), Emily R. Derbyshire(Duke University), Yvonne Van Gessel(Eisai (United States)), Sandra Duffy(Griffith University), Anne‐Marie Zeeman(Biomedical Primate Research Centre), Branko Mitasev(Eisai (United States)), Nicolas M. B. Brancucci(Swiss Tropical and Public Health Institute), Elizabeth A. Winzeler(University of California San Diego), Jeremy R. Duvall(Mersana Therapeutics (United States)), Amanda K. Lukens(Broad Institute), John E. Burke(University of Victoria), Sean Eckley(Eisai (United States)), Marshall Morningstar(Broad Institute), Takashi Yoshinaga(Eisai (Japan)), Fabian Gusovsky(Eisai (Japan)), Koen J. Dechering(TropIQ Health Sciences), Benito Muñoz(Broad Institute), Elamaran Meibalan(Harvard University)
Nature
September 7, 2016
Cited by 270


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