5′‐(<i>E</i>)‐Vinylphosphonate: A Stable Phosphate Mimic Can Improve the RNAi Activity of siRNA–GalNAc Conjugates

Rubina Parmar(Alnylam Pharmaceuticals (United States)), Vasant Jadhav(Alnylam Pharmaceuticals (United States)), Rachel Meyers(Alnylam Pharmaceuticals (United States)), Yi Pei(United States Military Academy), Donald J. Foster(Alnylam Pharmaceuticals (United States)), Laura Sepp‐Lorenzino(Intellia Therapeutics (United States)), Jennifer L. S. Willoughby(Alnylam Pharmaceuticals (United States)), Benjamin Brigham(Alnylam Pharmaceuticals (United States)), Martin A. Maier(Alnylam Pharmaceuticals (United States)), Walter Strapps, Christopher S. Theile(Alnylam Pharmaceuticals (United States)), Akin Akinc(Alnylam Pharmaceuticals (United States)), Muthiah Manoharan(Alnylam Pharmaceuticals (United States)), Kallanthottathil G. Rajeev(Alnylam Pharmaceuticals (United States)), Matthew G. Stanton(United States Military Academy), Jingxuan Liu(Alnylam Pharmaceuticals (United States)), Erin N. Guidry(Merck & Co., Inc., Rahway, NJ, USA (United States)), Klaus Charissé(Alnylam Pharmaceuticals (United States)), Mark T. Cancilla
ChemBioChem
April 28, 2016
Cited by 140


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