The discovery of 2-substituted phenol quinazolines as potent RET kinase inhibitors with improved KDR selectivity

Rebecca Newton(University of Manchester), Donald Ogilvie(Bioscience Research), Laura A. Maguire(University of Manchester), Daniel P. Mould(University of Manchester), Neil Q. McDonald(The Francis Crick Institute), Amanda Lyons(University of Manchester), H. Nikki March(University of Manchester), Gemma V. Hopkins(University of Manchester), Sarah V. Holt(Pharma Nord (United Kingdom)), Katherine A. Bowler(University of Manchester), Bohdan Waszkowycz(University of Manchester), Samantha Fritzl(University of Manchester), Andrew G. Purkiss(Cancer Research UK), Alexandra Stowell(University of Manchester), Emily M. Burns(Cancer Research UK), Allan M. Jordan(Signature Research (United States)), Ian D. Waddell(Charles River Laboratories (United Kingdom)), Emma Fairweather(University of Manchester), Kristin Goldberg(University of Manchester), P Chapman(University of Manchester), Stuart Jones(University of Manchester), Graeme Thomson(University of Manchester), Niall M. Hamilton(Ninewells Hospital), Amanda J. Watson(University of Manchester), Helen Small(University of Manchester)
European Journal of Medicinal Chemistry
January 29, 2016
Cited by 40


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