Synthesis and structure–activity relationships of 3,4-diaminocyclobut-3-ene-1,2-dione CXCR2 antagonists

J. Robert Merritt, Jianping Chao, Lynne Ozgur, Laura L. Rokosz, Tara M. Stauffer, Kingsley H. Nelson(United States Pharmacopeial Convention), Wei Wang(Capital Medical University), Ge Li(Anhui Medical University), Bernd Kaiser, John J. Baldwin(United States Pharmacopeial Convention), Adriane Schilling(United States Pharmacopeial Convention), Michael P. Dwyer, Arthur G. Taveras
Bioorganic & Medicinal Chemistry Letters
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