Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent

Giuseppe Campiani(University of Siena), Silvio Caccia(University of Siena), Giovanna Guiso(University of Siena), Anna Ramunno(University of Siena), Francesca Bolacchi(University of Siena), Ettore Novellino(Università Cattolica del Sacro Cuore), Elena Morelli(European Institute of Oncology), Silvio Spadari(University of Siena), Francesca Aiello(University of Siena), Giovanni Greco(University of Naples Federico II), Monica Fabbrini(University of Siena), Barbara Bongiovanni(University of Siena), M Capozzi(University of Siena), Antonio Garofalo(University of Siena), Giovanni Maga(Istituto di Genetica Molecolare), Stefano Marini(University of Rome Tor Vergata), Laura Ventura(University of Siena), Vito Nacci(University of Siena), Alberto Bergamini(University of Rome Tor Vergata), Silvia Armaroli(University of Siena)
Journal of Medicinal Chemistry
January 3, 2001
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