Inhibitors that stabilize a closed RAF kinase domain conformation induce dimerization
Hugo Lavoie(Defence Research and Development Canada), Marc Therrien(Institute for Research in Immunology and Cancer), Gwenaëlle Gavory(Institute for Research in Immunology and Cancer), Frank Sicheri(Mount Sinai Hospital), Jean Duchaine(Institute for Research in Immunology and Cancer), Michel Bouvier(University of California, San Francisco), Sébastien Guiral(Institute for Research in Immunology and Cancer), Neroshan Thevakumaran(Mount Sinai Hospital), John J. Li(Mount Sinai Hospital), Abbas Padeganeh, Daniel Y.L. Mao(Mount Sinai Hospital)
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