Bioactivation of 2,3-Diaminopyridine-Containing Bradykinin B<sub>1</sub> Receptor Antagonists: Irreversible Binding to Liver Microsomal Proteins and Formation of Glutathione Conjugates
Cuyue Tang, Thomayant Prueksaritanont(United States Military Academy), Ping Lü(Xiamen University), Scott D. Kuduk(Kettering University), Raju Subramanian(Gilead Sciences (United States)), Thomas A. Baillie(University of Washington), Eric D. Soli(Merck & Co., Inc., Rahway, NJ, USA (United States)), Sergey Krymgold, Mark G. Bock, Jonathan Z. Ho, Yuhsin Kuo, Dong-Mei Feng, Christina Ng(Orygen)
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