Catalysis of the CC-1065 and duocarmycin DNA alkylation reaction: DNA binding induced conformational change in the agent results in activation

Dale L. Boger(Scripps Research Institute), R. M. Garbaccio(Merck & Co., Inc., Rahway, NJ, USA (United States))
Bioorganic & Medicinal Chemistry
February 1, 1997
Cited by 89


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