BIOACTIVATION OF THE 3-AMINO-6-CHLOROPYRAZINONE RING IN A THROMBIN INHIBITOR LEADS TO NOVEL DIHYDRO-IMIDAZOLE AND IMIDAZOLIDINE DERIVATIVES: STRUCTURES AND MECHANISM USING 13C-LABELS, MASS SPECTROMETRY, AND NMRRaju Subramanian, Rominder Singh, Maria Victoria Silva Elipe et al.|Drug Metabolism and Disposition|2003Cited by 11
INDUCTION OF CYP1A IN THE BEAGLE DOG BY AN INHIBITOR OF KINASE INSERT DOMAIN-CONTAINING RECEPTOR: DIFFERENTIAL EFFECTS IN VITRO AND IN VIVO ON MRNA AND FUNCTIONAL ACTIVITYChristopher R. Gibson, Thomas H. Rushmore, Charles C. Lin et al.|Drug Metabolism and Disposition|2005Cited by 6