Tetrahydroindazoles as Interleukin-2 Inducible T-Cell Kinase Inhibitors. Part II. Second-Generation Analogues with Enhanced Potency, Selectivity, and Pharmacodynamic Modulation in VivoJason D. Burch, Zhonghua Pei, Charles Eigenbrot et al.|Journal of Medicinal Chemistry|2015Cited by 47
Enantioselective synthesis of GNE-6688, a potent and selective inhibitor of interleukin-2 inducible T-cell kinase (ITK)Jared T. Moore, Jason D. Burch, Kevin Lau et al.|Tetrahedron Letters|2019Cited by 3