Novel methyl substituted 1-(5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)methanones are P2X7 antagonists

Dale A. Rudolph(Janssen (United States)), Michael A. Letavic(Janssen (United States)), Michael K. Ameriks(Janssen (United States)), Pascal Bonaventure(Janssen (United States)), Nicholas I. Carruthers(Io Therapeutics (United States)), Hong Ao(Janssen (United States)), Anindya Bhattacharya(University of York), Meri De Angelis(Helmholtz Zentrum München), Christa C. Chrovian(Janssen (United States)), Jason C. Rech(Janssen (United States)), Brian Lord(Janssen (United States)), Qi Wang(Hebei Medical University), Ana B. Antón, José Ignacio Andrés, Jesús Alcázar(Janssen (Belgium))
Bioorganic & Medicinal Chemistry Letters
June 12, 2015
Cited by 33


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