Discovery of ARQ-501 as a potent PafA inhibitor that elevates KatG levels to potentiate isoniazid in mycobacteria

Cong Li(University of Electronic Science and Technology of China), Qingxiang Sun(University of Electronic Science and Technology of China), Hang Xiong(West China Medical Center of Sichuan University), Qiaohua Yan(University of Electronic Science and Technology of China), Cuiting Fang(Chinese Academy of Sciences), Bingzhou Huang(University of Electronic Science and Technology of China), Yan Liu(Sichuan University), Peng Xu(Shenzhen Third People’s Hospital), T Luo(West China Medical Center of Sichuan University), Youfu Luo(Sichuan University)
bioRxiv (Cold Spring Harbor Laboratory)
June 3, 2026
Cited by 0


Related Papers