Structure-Based Design of a Novel Covalent 4-(1-Methylindol-3-yl)pyrimidin-2-amine Series Targeting FGFR2 Resistance Mutations

Robert L. Hudkins(State Street (United States)), Daniel C. Bensen(State Street (United States)), Isaac Hoffman(Electronic BioSciences (United States)), Kirk Nelson(Arcturus Therapeutics (United States)), Alexandra Balcer(State Street (United States)), Melissa Neal(State Street (United States)), Ronald V. Swanson(Diversitech (United States)), Qing Ye(State Street (United States)), Todd J. Harris(State Street (United States)), Marc Rideout(State Street (United States)), Eric Allen(State Street (United States)), Samhita Iyer(State Street (United States)), Caleb B. Frye(State Street (United States)), Jacqueline H. Starrett(State Street (United States))
Journal of Medicinal Chemistry
March 31, 2026
Cited by 0


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