Two-Step Ligand-Directed Covalent Fluorescent Labeling of the Adenosine A <sub>1</sub> -Receptor That Maintains Its Orthosteric Binding Site’s Availability to Bind Ligands

Chia-Yang Lin(University of Nottingham), Stephen J. Hill(University of Nottingham), Joëlle Goulding(University of Nottingham), Barrie Kellam(University of Nottingham), Stephen J. Briddon(University of Nottingham), Simon Platt(University of Nottingham), Clare R. Harwood(University of Nottingham), Chih-Wei Lai(National Defense University), Nicholas D. Kindon(University of Nottingham)
Journal of Medicinal Chemistry
January 8, 2026
Cited by 0


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