Discovery of DS79540454 via fragment-based drug discovery strategy: New scaffolds of hypoxia-inducible factor prolyl hydroxylase inhibitor

Takeshi Fukuda(Jikei University School of Medicine), Naoki Tanaka(Kyushu University), Y. Kawabata(Daiichi-Sankyo (Japan)), Ken J. Ishii(The University of Tokyo), Shinichi Takahashi(Daiichi-Sankyo (Japan)), Daichi Baba(Yokohama City University), Shuichiro Ito(Daiichi-Sankyo (Japan)), Tatsuya Nishi(Okayama University), Kyoji Yamaguchi(Daiichi-Sankyo (Japan)), Takashi Ishiyama(Daiichi-Sankyo (Japan)), Riko Kitazawa(Ehime University Hospital)
Bioorganic & Medicinal Chemistry Letters
November 20, 2025
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