Topobexin Targets a Unique Druggable Pocket of Topoisomerase II for Beta Isoform- Selective Control of DNA Damage During Anthracycline Chemotherapy

Jan Kubeš(University Hospital Hradec Králové), Matthew J. Schellenberg(Mayo Clinic), Anna Jirkovská(University Hospital Hradec Králové), Galina Karabanovich(University Hospital Hradec Králové), Taylor L. Witter(Mayo Clinic), Caroline A. Austin(Newcastle University), Iuliia Melnikova(University Hospital Hradec Králové), Veronika Keresteš(University Hospital Hradec Králové), Olga Lencova(University Hospital Hradec Králové), Anh Cong(Mayo Clinic in Arizona), Hana Bavlovic Piskackova(University Hospital Hradec Králové), Petra Štěrbová‐Kovaříková(University Hospital Hradec Králové), Tomáš Šimůnek(Charles University), Jaroslav Roh(Charles University), Martin Štěrba(Charles University), Lenka Applová(University Hospital Hradec Králové), Jasmina Paluncic, Jiřı́ Kuneš(University Hospital Hradec Králové), Julia R Alvey(Mayo Clinic in Arizona), Lise C. M. Arrouye(Mayo Clinic in Arizona), Petra Kollárová-Brázdová(University Hospital Hradec Králové)
Structural Dynamics
September 1, 2025
Cited by 0


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