Single-Dose Oral Influenza Antiviral Prodrug Enabled by Cholesterol Conjugation

Chenning Li(Chinese Academy of Sciences), Xuebing Li(Tianjin Medical University General Hospital), Lifeng Fu(Chinese Academy of Sciences), Yiran Li(Chinese Academy of Medical Sciences & Peking Union Medical College), Shuihong Cheng(Chinese Academy of Sciences), Chenxi Cheng(Shenyang Pharmaceutical University), Yuhai Bi(Chinese Academy of Sciences), Xun Lv(Chinese Academy of Sciences), George F. Gao(Chinese Academy of Sciences)
Journal of Medicinal Chemistry
October 3, 2025
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