Enantioselective β-C(sp <sup>3</sup> )–H Nucleophilic Tosylation of Native Amides: A Synthetic Platform for Chiral Methyl Stereocenters

Yuxin Ouyang(Scripps Research Institute), Jin‐Quan Yu(Scripps Research Institute), Yi-Hao Li(Scripps Research Institute), Nikita Chekshin(Scripps Research Institute), Jennifer X. Qiao(Princeton University), D. Quang Phan(Scripps Research Institute), Martin D. Eastgate(Bristol-Myers Squibb (United States))
Journal of the American Chemical Society
May 31, 2025
Cited by 12


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