Abstract 4231: Preclinical candidate RVU305, an MTA-cooperative PRMT5 inhibitor, shows activity in MTAP-deleted tumors resistant to immune checkpoint treatment
Anna Bartosik, Krzysztof Brzózka, Tomasz Rzymski, Jacek Faber, Beata Kowalska(Lublin University of Technology), Mateusz Stoszko(Erasmus MC), Michał Combik, Jacek Stępniewski, Bożena Winnik, Marta Wadowska, Aleksandra Więckowska, Agnieszka Szymula, Kamil Kuś, Paulina Podkalicka(Jagiellonian University), Aneta Bobowska(Medical University of Warsaw), Karolina Gluza, Agnieszka H. Ludwig‐Słomczyńska(Jagiellonian University), Mateusz Ogórek, Stefan Chmielewski, Mateusz Nowak, Kamila Białkowska, Joanna Krawczyk, Maciej Kujawa, Oleksii Bryzghalov, Marcin Kowiel, Adam Radzimierski, Kamila Kozłowska-Tomczyk(Jagiellonian University), Milena Mazan(Wellcome Sanger Institute), Lika Osugui, Szymon Woroszyło, Aniela Gołas, Didier Pez, Agata Stachowicz-Wałaszek, Adrian Zarębski(Jagiellonian University), Julia Wirkijowska, Agnieszka Piątek
Cited by 1
Related Papers
A CRISPR Dropout Screen Identifies Genetic Vulnerabilities and Therapeutic Targets in Acute Myeloid Leukemia
|Cell Reports|2016|834
The Role of ATF4 Stabilization and Autophagy in Resistance of Breast Cancer Cells Treated with Bortezomib
|Cancer Research|2009|298
Role of ATF4 in regulation of autophagy and resistance to drugs and hypoxia
|Cell Cycle|2009|197
Gfi1 Coordinates Epigenetic Repression of <i>p21</i><sup><i>Cip/WAF1</i></sup> by Recruitment of Histone Lysine Methyltransferase G9a and Histone Deacetylase 1
|Molecular and Cellular Biology|2005|170
Hypoxic activation of the unfolded protein response (UPR) induces expression of the metastasis-associated gene LAMP3
|Radiotherapy and Oncology|2009|98