Alkyl Sulfonylhydrazide-Enabled, Chemoselective Ni-catalyzed Directed C(sp2)–H Alkylation via Low-Temperature, Amine-Assisted Metalation/Deprotonation

Shuanghu Wang, Keary M. Engle(Scripps Research Institute), Yilin Cao(Scripps Research Institute), Yu Kawamata(Scripps Research Institute), David A. Cagan(California Institute of Technology), Maximilian D. Palkowitz(Bristol-Myers Squibb (Germany)), Benjamin Vokits(Bristol-Myers Squibb (United States)), Phil S. Baran(Scripps Research Institute)
ChemRxiv
March 25, 2025
Cited by 7


Related Papers