Developing potent anti-inflammatory IRAK4-targeting PROTACs with simplified CRBN ligands
Yu Rao(Soochow University), Peilu Song(Tsinghua University), Yujie Liu(Shanxi University of Traditional Chinese Medicine), Xiuyun Sun(Tsinghua University), Xin Zhai(Shenyang Pharmaceutical University)
Cited by 2
Related Papers
PROTACs: great opportunities for academia and industry
|Signal Transduction and Targeted Therapy|2019|627
PROTAC Technology: Opportunities and Challenges
|ACS Medicinal Chemistry Letters|2020|353
PROTAC-induced BTK degradation as a novel therapy for mutated BTK C481S induced ibrutinib-resistant B-cell malignancies
|Cell Research|2018|280
Chemistries of bifunctional PROTAC degraders
|Chemical Society Reviews|2022|270