Discovery of Covalent and Cell‐Active ALKBH5 Inhibitors with Potent Antileukemia Effects <i>In Vivo</i>

Hengbo Wu(Tongji University), Gan‐Qiang Lai(Saint Louis University), Chunpu Li(Chinese Academy of Sciences), Hui Huang(Chinese Academy of Sciences), Jing Gao(Chinese Academy of Sciences), Hu Zhou, Ruixiang Cheng(Chinese Academy of Sciences), Zeyu Liu(Chinese Academy of Sciences), Cai‐Guang Yang(Shanghai Jiao Tong University), Ju Wang(Chinese Academy of Sciences)
Angewandte Chemie
February 20, 2025
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