Exploring Alternative Zinc-Binding Groups in Histone Deacetylase (HDAC) Inhibitors Uncovers <b>DS-103</b> as a Potent Ethylhydrazide-Based HDAC Inhibitor with Chemosensitizing Properties

Daniel Stopper(University of Bonn), Finn K. Hansen(University of Bonn), Linda Schäker‐Hübner(University of Bonn), Beate König(University of Bonn), P. R. Watson(Johns Hopkins University), Jingyu Li(Heinrich Heine University Düsseldorf), Jana Klose(Canada's Michael Smith Genome Sciences Centre), Daniel Ramsbeck(Anhalt University of Applied Sciences), Alexandra Hamacher(Heinrich Heine University Düsseldorf), Matthias U. Kassack(Heinrich Heine University Düsseldorf), Maria Hanl(University of Bonn), Laís Pessanha de Carvalho(Research Institute for Tropical Medicine), Matthew N. Gaynes(University of Pennsylvania), Jana Held(Research Institute for Tropical Medicine), Lukas Biermann(Heinrich Heine University Düsseldorf), David W. Christianson(California University of Pennsylvania)
Journal of Medicinal Chemistry
February 13, 2025
Cited by 12


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