Optimization of Single Relaxin B-Chain Peptide Leads to the Identification of R2R01, a Potent, Long-Acting RXFP1 Agonist for Cardiovascular and Renal Diseases

Sergio Mallart(Sanofi (France)), Stéphane Illiano(Délégation Paris 5), Laura Orsatti(IRBM Science Park), Alain Corbier(Sanofi (France)), Xavier Chénedé(Sanofi (France)), Frank Marguet(Sanofi (France)), Daniela Roversi(IRBM Science Park), Claire Minoletti(Sanofi (France)), Denis Brasseur(Sanofi (France)), Bernard Maillère(Commissariat à l'Énergie Atomique et aux Énergies Alternatives), Olivier Duclos(Sanofi (France)), Edith Monteagudo(IRBM Science Park), Bruno Poirier(Sanofi (France)), Fulvia Caretti(IRBM Science Park), Annalise Di Marco(IRBM Science Park), Laurence Gauzy‐Lazo(Sanofi (France)), Aurélien Azam(Commissariat à l'Énergie Atomique et aux Énergies Alternatives), Maria Veneziano(IRBM Science Park), Raffaele Ingenito, Elisabetta Bianchi(IRBM Science Park), Alessia Santoprete(IRBM Science Park), Vincent Gervat(Sanofi (France)), Alberto Bresciani(University of Bergamo), Paola Magotti(IRBM Science Park), Simone Esposito(IRBM Science Park), Olivier Pasquier(Sanofi (France)), Philip Janiak(Hôpital Lariboisière)
Journal of Medicinal Chemistry
January 31, 2025
Cited by 1


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