Chemoproteomic discovery of a covalent allosteric inhibitor of WRN helicase
Kristen A. Baltgalvis(Vividion Therapeutics (United States)), Kelsey N. Lamb(Vividion Therapeutics (United States)), Kent T. Symons(Vividion Therapeutics (United States)), Chu-Chiao Wu(Vividion Therapeutics (United States)), Melissa Hoffman(Vividion Therapeutics (United States)), Aaron N. Snead(Vividion Therapeutics (United States)), Xiaodan Song(Vividion Therapeutics (United States)), Thomas Glaza(Vividion Therapeutics (United States)), Shota Kikuchi(Vividion Therapeutics (United States)), Jason C. Green(Vividion Therapeutics (United States)), Donald C. Rogness(Vividion Therapeutics (United States)), Betty Lam(Vividion Therapeutics (United States)), Maria E. Rodriguez-Aguirre(Vividion Therapeutics (United States)), David R. Woody(Vividion Therapeutics (United States)), Christie L. Eissler(Vividion Therapeutics (United States)), Socorro Rodiles(Vividion Therapeutics (United States)), Seth M. Negron(Vividion Therapeutics (United States)), Steffen M. Bernard(Vividion Therapeutics (United States)), Eileen Tran(Vividion Therapeutics (United States)), Jonathan Pollock(Vividion Therapeutics (United States)), Ali Tabatabaei(Vividion Therapeutics (United States)), Víctor Contreras(Vividion Therapeutics (United States)), Heather N. Williams(Vividion Therapeutics (United States)), Martha K. Pastuszka(Vividion Therapeutics (United States)), J. Sigler(Vividion Therapeutics (United States)), Piergiorgio Pettazzoni(Roche (Switzerland)), M.G. Rudolph(Roche (Switzerland)), Moritz Classen(Roche (Switzerland)), Doris Brugger(Roche (Switzerland)), Christopher F. Claiborne(Roche (Switzerland)), Jean‐Marc Plancher(Roche (Switzerland)), Isabel Cuartas(Universitat Autònoma de Barcelona), Joan Seoane(Universitat Autònoma de Barcelona), Laurence E. Burgess(Vividion Therapeutics (United States)), Robert T. Abraham(Vividion Therapeutics (United States)), David S. Weinstein(Vividion Therapeutics (United States)), Gabriel M. Simon(Vividion Therapeutics (United States)), Matthew P. Patricelli(Vividion Therapeutics (United States)), Todd M. Kinsella(Vividion Therapeutics (United States))
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