Discovery of a Novel Thienopyrimidine Compound as a Urate Transporter 1 and Glucose Transporter 9 Dual Inhibitor with Improved Efficacy and Favorable Druggability

Xiaoyu Shi(Shandong University), Peng Zhan(Shandong University of Traditional Chinese Medicine), Fengxin Zheng(Southern Medical University), Ming‐Yu Yang(The Affiliated Yongchuan Hospital of Chongqing Medical University), Zhenqian Wang(Stockholm University), Youzhao Wang(Northeastern University), Xinyong Liu(Shandong University of Traditional Chinese Medicine), Jianxin Pang(Southern Medical University), Shenghua Gao, Shuo Wang(Jiangnan University), Jian Zhang(Shandong University), Shujing Xu(Shandong University), Hui Liao(Huazhong University of Science and Technology), Zhen Gao(Shandong University), Fan Yi(Shandong University), Qian Yang, Danhui Qi(Shandong University), Tong Zhao(China Pharmaceutical University), Zhijiao Zhang(Shandong University of Traditional Chinese Medicine)
Journal of Medicinal Chemistry
March 14, 2024
Cited by 16


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