Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
Ning Zhuo(Chinese Academy of Sciences), Fajun Nan(Chinese Academy of Sciences), Shimeng Guo(Shanghai Institute of Materia Medica), Min Gu(Chinese Academy of Sciences), Chenlu Zhang(Northwestern University), Tingting Zhao(Northeastern University), Jianpeng Yin(Ministry of Agriculture and Rural Affairs), Xiu Run Ge(Chinese Academy of Sciences), Ying Yun(Shanghai Institute of Materia Medica), Xin Xie(Binzhou Medical University)
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