Co-opting the E3 ligase KLHDC2 for targeted protein degradation by small molecules

Christopher M. Hickey(Arvinas (United States)), Katherine M. Digianantonio(Arvinas (United States)), Kurt Zimmermann(Arvinas (United States)), Alicia Harbin(Arvinas (United States)), Connor Quinn(Arvinas (United States)), Avani Patel(Arvinas (United States)), Peter C. Gareiss(Arvinas (United States)), Amanda Chapman(Arvinas (United States)), Bernadette Tiberi(Thomas Jefferson University), Jennifer Dobrodziej(Accent Therapeutics (United States)), John Corradi(Arvinas (United States)), Angela Cacace(Arvinas (United States)), David R. Langley(Arvinas (United States)), Miklós Békés(Arvinas (United States))
Nature Structural & Molecular Biology
January 4, 2024
Cited by 58

Abstract


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