Structure-Based Discovery of a NPFF1R Antagonist with Analgesic Activity
Brian J. Bender(University of California, San Francisco), Brian K. Shoichet(University of California, San Francisco), Bryan L. Roth(University of North Carolina at Chapel Hill), Hye Jin Kang(University of North Carolina at Chapel Hill), Stefan Gahbauer(University of California, San Francisco), Julie E. Pickett(University of North Carolina at Chapel Hill), Karnika Bhardwaj(University of California, San Francisco), João M. Bráz(University of California, San Francisco), Yongfeng Liu(University of North Carolina at Chapel Hill), Sian Rodriguez-Rosado(Universidad Católica de Santa Fe), Manish K. Jain(University of North Carolina at Chapel Hill), Allan I. Basbaum(W. M. Keck Foundation)
Cited by 5
Related Papers
The promise and peril of chemical probes
|Nature Chemical Biology|2015|848
4-Hydroxynonenal, an endogenous aldehyde, causes pain and neurogenic inflammation through activation of the irritant receptor TRPA1
|Proceedings of the National Academy of Sciences|2007|762
A practical guide to large-scale docking
|Nature Protocols|2021|540
Dorsal root ganglion macrophages contribute to both the initiation and persistence of neuropathic pain
|Nature Communications|2020|515
Peptides and the primary afferent nociceptor
|Journal of Neuroscience|1993|484