Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia

Jingyu Zhang(Hangzhou First People's Hospital), Jinxin Che(Second Affiliated Hospital of Zhejiang University), Shenxin Zeng(Hangzhou Medical College), Wenhai Huang(Hangzhou Medical College), Nengming Lin(Hangzhou First People's Hospital), Ao Pang(Zhejiang University), Yuheng Jin(Zhejiang University), Yubo Zhou(Shanghai Institutes for Biological Sciences), Yuwei Wang(Shanghai Jiao Tong University), Haiting Duan(Zhejiang University), Xiaoli Yu(Zhejiang University), Xiaojun Yao(Quality Research), Mingfei Wu(Zhejiang Institute of Mechanical and Electrical Engineering), Jia Li(Shanghai Institute of Materia Medica), Liteng Shen(Zhejiang Lab), Renzhao Gui(Zunyi Medical University), Bo Zhang(Hangzhou First People's Hospital), Xiaowu Dong(Zhejiang University)
European Journal of Medicinal Chemistry
October 17, 2023
Cited by 14


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