Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia

Jingyu Zhang(Hangzhou First People's Hospital), Jinxin Che(Pharmaceutical Biotechnology (Czechia)), Shenxin Zeng(Hangzhou Medical College), Wenhai Huang(Hangzhou Medical College), Nengming Lin(Westlake University), Ao Pang(Zhejiang University), Yuheng Jin(Zhejiang University), Yubo Zhou(Sichuan Mianyang 404 Hospital), Yuwei Wang(Peking University), Haiting Duan(Zhejiang University), Xiaoli Yu(Zhejiang University), Xiaojun Yao(Macau University of Science and Technology), Mingfei Wu(Zhejiang University), Jia Li(Shanghai Institute of Materia Medica), Liteng Shen(Zhejiang Lab), Renzhao Gui(Zunyi Medical University), Bo Zhang(Hangzhou First People's Hospital), Xiaowu Dong(Second Affiliated Hospital of Zhejiang University)
European Journal of Medicinal Chemistry
October 17, 2023
Cited by 14


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